Stimulants

G-130

Summary G-130 (also known as GP-130 or 2-Phenyl-5,5-dimethyltetrahydro-1,4-oxazine) is a pharmaceutical compound recognized for its stimulant and anorectic properties, and it shares a chemical relationship with phenmetrazine. Identifiers IUPAC name CAS Number 42013-48-9  PubChem CID 97711 ChemSpider 88190 UNII 785F2C727T CompTox Dashboard (EPA) DTXSID40963342 Chemical and physical data Formula C12H17NO Molar mass 191.274 g·mol−1 Synthesis Ex …

G-130 Read More »

2-Phenyl-3,6-dimethylmorpholine

Summary 2-Phenyl-3,6-dimethylmorpholine, a pharmaceutical compound, is known for its stimulant and anorectic properties and is closely associated with phenmetrazine. With structural similarities to other phenylmorpholine compounds, it is believed to function as a serotonin reuptake inhibitor, potentially yielding effects akin to antidepressants. Nonetheless, anecdotal accounts propose that its activity primarily involves inducing anorectic effects, with …

2-Phenyl-3,6-dimethylmorpholine Read More »

4-Methylphenmetrazine

Summary 4-Methylphenmetrazine, also known as mephenmetrazine, 4-MPM, or PAL-747, is a recreational designer substance celebrated for its stimulating effects. This compound is a derivative of phenylmorpholine, sharing a close structural relation with more widely recognized substances like phenmetrazine and 3-fluorophenmetrazine. It initially came to attention in Slovenia in 2015, and subsequent research has revealed its …

4-Methylphenmetrazine Read More »

4′-Fluoro-4-methylaminorex

Summary 4′-Fluoro-4-methylaminorex, commonly called 4F-MAR or 4-FPO, is a recreational designer drug from the substituted aminorex class. This compound is known for its stimulant properties. Its presence was initially identified in Slovenia in the year 2018. Notably, it was subjected to legal prohibition in Italy in March 2020. Identifiers IUPAC name CAS Number 1364933-64-1  PubChem …

4′-Fluoro-4-methylaminorex Read More »

Propylphenidate

Summary Propylphenidate, sometimes called PPH, belongs to the class of piperidine-based stimulant drugs. It shares a close structural relationship with methylphenidate, differing primarily in replacing the methyl ester with a propyl ester. Notably, in April 2015, the United Kingdom classified Propylphenidate as a Temporary Class Drug due to its unauthorized distribution and sale as a …

Propylphenidate Read More »

Meprylcaine

Summary Meprylcaine, also known as Epirocaine and Oracaine, is a local anesthetic featuring stimulant characteristics and shares a structural resemblance with dimethocaine.This compound boasts a noteworthy capacity to inhibit monoamine transporters, effectively impeding the reuptake of crucial neurotransmitters such as dopamine, norepinephrine, and serotonin. Identifiers IUPAC name CAS Number 495-70-5 PubChem CID 4065 ChemSpider 3925 …

Meprylcaine Read More »

Benocyclidine

Summary Benocyclidine, also recognized as benzo​thiophenyl​cyclo​hexylpiperidine (BTCP), represents a psychoactive recreational substance within the arylcyclohexylamine class, closely associated with phencyclidine (PCP). The initial documentation of this compound can be traced back to a patent application submitted by Marc Caron and a team at Duke University in 1997.This potent and selective dopamine reuptake inhibitor (DRI) substance …

Benocyclidine Read More »

4-Methylmethylphenidate

Summary Threo-4-methylmethylphenidate (4-MeTMP) is a stimulant drug with a chemical relationship with methylphenidate. While it is akin to methylphenidate, its stimulant properties are somewhat milder, and it exhibits relatively limited effectiveness in inhibiting dopamine reuptake despite its high binding affinity. This unique profile has prompted investigations into its potential use as an alternative treatment for …

4-Methylmethylphenidate Read More »

Thiothinone

Summary Thiothinone, also known as βk-MPA, is a stimulant classified as the beta-keto substituted counterpart of methiopropamine. It has gained popularity as a designer drug and has been available for purchase on online platforms. Structurally, Thiothinone resembles methcathinone, except that the phenyl group has been replaced by a thiophene group.Interestingly, Thiothinone has also been identified …

Thiothinone Read More »

5-Methylmethiopropamine

Summary 5-Methylmethiopropamine (5-MMPA), or mephedrene, is a stimulant drug. Unlike mephedrone, it is not a substituted cathinone derivative because it lacks a ketone group at the β position of the aliphatic side chain. Instead, it bears a closer resemblance to substituted amphetamines. This compound was discovered in Germany in June 2020 and has since been …

5-Methylmethiopropamine Read More »