Summary RCS-4, also known as 1-pentyl-3-(4-methoxybenzoyl)indole, is a synthetic cannabinoid compound that has been marketed and sold under various names, including SR-19, BTM-4, Eric-4 (later abbreviated to E-4), and initially, OBT-199. Identifiers IUPAC name CAS Number 1345966-78-0 ChemSpider 24769418 UNII…
Summary AM-2233 is a pharmaceutical compound recognized for its exceptional role as a potent full agonist for cannabinoid receptors. Specifically, the (R) enantiomer of AM-2233 exhibits a remarkable Ki of 1.8 nM at CB1 and 2.2 nM at CB2, underscoring…
Summary AM-1241, also known as 1-(methylpiperidin-2-ylmethyl)-3-(2-iodo-5-nitrobenzoyl)indole, is a member of the aminoalkylindole family, recognized for its role as a potent and highly selective agonist for the cannabinoid receptor CB2. With a remarkable Ki value of 3.4 nM at CB2, it…
Summary AM-694, known chemically as 1-(5-fluorophenyl)-3-(2-iodobenzoyl)indole, functions as a designer drug with a specific role as a potent and selective agonist for the cannabinoid receptor CB1. This compound is frequently utilized in scientific research to map the distribution of CB1…
Summary AM-679, a member of the AM cannabinoid series, is a moderately potent agonist for cannabinoid receptors. It exhibits a Ki of 13.5 nM at CB1 and 49.5 nM at CB2, signifying its affinity for these receptors. Notably, AM-679 was…
Summary AM-630, or 6-Iodopravadoline, is a potent and highly selective inverse agonist targeting the cannabinoid receptor CB2. It exhibits a remarkable affinity for CB2, boasting a Ki value of 32.1 nM, while showing a notable 165-fold selectivity over CB1 receptors,…
